Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_01964
Ion Channel
Voltage-gated proton channel (Hv1)
Peptide Function
Inhibitor
Gene Name
HVCN1
Activity Data (nM)
IC50
Not available
Ki
1 nM
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
SSTCIPSGQPCADSDDCCETFHCKWVFFTSKFMCRRVWGKD
Peptide UniProt Accession
Not available
UniParc
UPI000F706501
Peptide Synonyms/Alias
Corza6
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
pH 7.5
Holding Potential (mV)
−50 mV
Temperature
Room Temperture
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Extracellular domain
Binding Site Residue
C6 appears to be specific to hHv1 since it does not cross-react with exemplar potassium and sodium VGICs (Voltage-gated potassium channel subfamily B member 1 and Sodium channel protein type 4 subunit alpha), CiHv1, or Catsper in Homo sapiens sperm
Ion Channel Information
Gene Abbreviation (ABB)
VGHC
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available